3108-27-8Relevant academic research and scientific papers
A tandem [3+2] cycloaddition-elimination cascade reaction to generate pyrrolo-[3,4-c]pyrrole-1,3-diones
Martinez-Ariza, Guillermo,Dietrich, Justin,De Moliner, Fabio,Hulme, Christopher
, p. 1801 - 1804 (2013/09/12)
An efficient tandem [3+2] cycloaddition-elimination cascade sequence has been developed enabling assembly of the pharmacologically relevant pyrrolo-[3,4-c]pyrrole-1,3-dione chemotype. The strategy involves simple mixing of readily accessible oxazolin-2-on
Application of a novel [3+2] cycloaddition reaction to prepare substituted imidazoles and their use in the design of potent DFG-out allosteric B-Raf inhibitors
Dietrich, Justin,Gokhale, Vijay,Wang, Xiadong,Hurley, Laurence H.,Flynn, Gary A.
experimental part, p. 292 - 304 (2010/04/02)
B-Raf protein kinase, which is a key signaling molecule in the RAS-RAF-MEK-ERK signaling pathway, plays an important role in many cancers. The B-Raf V600E mutation represents the most frequent oncogenic kinase mutation known and is responsible for increas
