31230-44-1Relevant articles and documents
A two step route to indoles from haloarenes - A versatile variation on the Fischer indole synthesis
Inman, Martyn,Moody, Christopher J.
, p. 788 - 790 (2011)
In a new variation on the Fischer indole synthesis, readily available haloarenes are converted into a wide range of indoles in just two steps by halogen-magnesium exchange, quenching with di-tert-butyl azodicarboxylate, followed by reaction with ketones u
Ruthenium-catalyzed synthesis of indoles from anilines and epoxides
Pena-Lopez, Miguel,Neumann, Helfried,Beller, Matthias
supporting information, p. 1818 - 1824 (2014/03/21)
A general synthetic route to indoles from readily available anilines and epoxides by using ruthenium catalysis is described. This straightforward transformation allows a variety of indoles to be obtained in good yields by using [Ru3(CO)12]/1,1-bis(diphenylphosphino)ferrocene as the catalytic system. Water and hydrogen are formed as the only stoichiometric by-products, making this process highly atom efficient.
Two-step route to indoles and analogues from haloarenes: A variation on the Fischer indole synthesis
Inman, Martyn,Carbone, Anna,Moody, Christopher J.
experimental part, p. 1217 - 1232 (2012/03/26)
In a new variation on the Fischer indole synthesis, readily available haloarenes are converted into a wide range of indoles in just two steps by halogen-magnesium exchange and quenching with di-tert-butyl azodicarboxylate, followed by reaction with aldehy
