32445-29-7Relevant articles and documents
Synthesis and biological characterization of amidopropenyl hydroxamates as HDAC inhibitors
Thaler, Florian,Varasi, Mario,Colombo, Andrea,Boggio, Roberto,Munari, Davide,Regalia, Nickolas,Rozio, Marco G.,Reali, Veronica,Resconi, Anna E.,Mai, Antonello,Gagliardi, Stefania,Dondio, Giulio,Minucci, Saverio,Mercurio, Ciro
experimental part, p. 1359 - 1372 (2011/01/12)
A series of amidopropenyl hydroxamic acid derivatives were prepared as novel inhibitors of human histone deacetylases (HDACs). Several compounds showed potency at 50 values in tests again