32445-29-7Relevant academic research and scientific papers
Synthesis and biological characterization of amidopropenyl hydroxamates as HDAC inhibitors
Thaler, Florian,Varasi, Mario,Colombo, Andrea,Boggio, Roberto,Munari, Davide,Regalia, Nickolas,Rozio, Marco G.,Reali, Veronica,Resconi, Anna E.,Mai, Antonello,Gagliardi, Stefania,Dondio, Giulio,Minucci, Saverio,Mercurio, Ciro
experimental part, p. 1359 - 1372 (2011/01/12)
A series of amidopropenyl hydroxamic acid derivatives were prepared as novel inhibitors of human histone deacetylases (HDACs). Several compounds showed potency at 50 values in tests again
Heterocyclic derivatives as HDAC inhibitors
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Page/Page column 15, (2009/12/27)
This invention is related to new histone deacetylase inhibitors according to the general formula (I) wherein: the dotted line is an optional additional bond; R1 is hydrogen, halogen, C1-C6 alkyl, C1-C6/sub
