33920-36-4Relevant academic research and scientific papers
Benzodiazepine derivatives, compositions containing them and their use in therapy
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, (2008/06/13)
Compounds of formula (I), and salts and prodrugs thereof STR1 wherein: R 1 is H, certain optionally substituted C 1.6 alkyl, or C 3-7 cycloalkyl;R 2 is (CH 2) q -tetrazolyl optionally substituted in the tetrazole ring by C 1-4 alkyl, (CH 2) q -imidazolyl
CHOLECYSTOKININ ANTAGONISTS
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, (2008/06/13)
Benzodiazepine analogs of the formula: STR1 are disclosed which are antagonists of gastrin and cholecystokinin (CCK).
Benzodiazepine derivatives, compositions containing them and their use in therapy
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, (2008/06/13)
Compounds of formula (I), and salts and prodrugs thereof wherein: R1 represents optionally substituted C? ??alkyl or C???cycloalkyl; R2 represents an optionally substituted phenyl or pyridyl group; R3 represents C??? alkyl or halo; R? represents C??? cycloalkyl; X is 0, 1, 2 or 3; are CCK and/or gastrin antagonists. They and compositions thereof are therefore useful in therapy.
