34491-79-7Relevant articles and documents
Refining the structure?activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms
Magalh?es, Joana,Franko, Nina,Annunziato, Giannamaria,Pieroni, Marco,Benoni, Roberto,Nikitjuka, Anna,Mozzarelli, Andrea,Bettati, Stefano,Karawajczyk, Anna,Jirgensons, Aigars,Campanini, Barbara,Costantino, Gabriele
, p. 31 - 43 (2018/11/01)
The lack of efficacy of current antibacterials to treat multidrug resistant bacteria poses a life-threatening alarm. In order to develop enhancers of the antibacterial activity, we carried out a medicinal chemistry campaign aiming to develop inhibitors of