356039-77-5Relevant academic research and scientific papers
Facile synthesis of 7-10 membered rings by intramolecular condensation using dialkylcarbonate as solvent
Ikemoto, Tomomi,Ito, Tatsuya,Nishiguchi, Atsuko,Tomimatsu, Kiminori
, p. 9335 - 9339 (2007/10/03)
A convenient large-scalable synthesis of 1-benzazepines 19 as an important intermediate of CCR5 antagonist, oral HIV-1 therapy, was established. The anilination of o-halogenobenzaldehyde 9 with alkylamino-acid 16 gave o-formylaniline-acid 17. Compound 17
Process for producing cyclic compound
-
, (2008/06/13)
A process suitable for safely mass-producing, through a short step, cyclic compounds useful in medicines, agricultural chemicals, foods, cosmetics, and chemical products or as intermediates therefor. The process, which is for producing a compound represen
