361531-79-5Relevant academic research and scientific papers
A Flexible Approach for the Asymmetric Synthesis of N-Protected (R) -5-Alkyl Tetramates and (R)-5-Alkyl Tetramic Acid Derivatives
Huang, Pei-Qiang,Deng, Jun
, p. 247 - 250 (2007/10/03)
A flexible two-step asymmetric approach to N-protected (R)-5-alkyl tetramates and (R)-5-alkyl tetramic acid derivatives is described. The method is based on the diastereoselective alkylation of (R)-phenylglycinol derived tetramates 7 and 8, which are the
SUBSTITUTED PIPERODINES AND PYRROLIDINES AS CALCIUM SENSING RECEPTOR MODULATORS AND METHOD
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Page 35, (2008/06/13)
Compounds are provided which are antagonists of the calcium sensing receptor, and have the general formula (I) wherein m is 0, 1, 2, 3 or 4; each X is independently selected from the group consisting of hydrogen, halo, cyano, nitro, OCF3, hydroxy, amino,
Design of potential new HIV protease inhibitors: Enantioconvergent synthesis of new pyrrolidin-3-ol, and pyrrolidin-3-one peptide conjugates
Courcambeck,Bihel,De Michelis,Quelever,Kraus
, p. 1421 - 1430 (2007/10/03)
Novel potential HIV protease inhibitors are obtained by an enantioconvergent synthesis of mimicking Phe-Pro dipeptides, achieved through the coupling between Boc(L)Phe or Boc(L)Tyr and both enantiomers of syn-2-benzylpyrrolidin-3-ol and their correspondin
