36374-63-7Relevant academic research and scientific papers
Aza vinyl sulfones: Synthesis and evaluation as antiplasmodial agents
Glória, Paulo M.C.,Gut, Jiri,Gonalves, Lídia M.,Rosenthal, Philip J.,Moreira, Rui,Santos, Maria M.M.
scheme or table, p. 7635 - 7642 (2012/01/05)
A series of novel aza vinyl sulfones were designed, synthesized in good yields and evaluated as antiplasmodial agents. Tested compounds did not show activity against papain or the Plasmodium falciparum cysteine protease falcipain-2. However, a number of t
Modified amino acids
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Page/Page column 11, (2008/06/13)
The present invention provides a compound of the general formula 1, wherein X is the connection between the CO-hydrazine and the NR1-oxalic acid or ester group, and uses and synthesis methods. These compounds represent amino acid derivatives, wherein the amine group is turned into an acidic group by the oxalic acid group and the carboxylic acid is turned into an amine functionality by the hydrazine group; as well as peptidomimetics comprising the compound and methods for their synthesis.
