364607-96-5

Upstream product

• 5339-85-5 2-aminophenethyl alcohol 
• 155164-66-2 2-benzoyl-4,5-dichloropyridazin-3(2H)-one 
• 98-88-4 benzoyl chloride 
• 869469-13-6 trifluoro-methanesulfonic acid 2-(2-hydroxy-ethyl)-phenyl ester 
• 869469-11-4 trifluoro-methanesulfonic acid 2-(2-oxo-ethyl)-phenyl ester 
• 109586-43-8 o-(2-propenyl)phenyl trifluoromethanesulfonate 
• 1745-81-9 o-Allylphenol 
• 869468-95-1 trifluoro-methanesulfonic acid 2-[2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-phenyl ester 

Downstream Products

• 61589-14-8 N-benzoylindoline 
• 860521-17-1 benzoic acid-[2-(2-chloro-ethyl)-anilide] 
• 869468-74-6 carbonic acid 2-(2-benzoylamino-phenyl)-ethyl ester methyl ester 
• 175846-71-6 N-(2-vinyl-phenyl)benzamide 

Relevant academic research and scientific papers

A domino amidation route to indolines and indoles: Rapid syntheses of anhydrolycorinone, hippadine, oxoassoanine, and pratosine

(Chemical Equation Presented) When subjected to palladium-catalyzed amidation conditions, 2-triflyloxy phenethyl carbonates undergo, in addition to the expected aryl cross-coupling, an additional amidation with net displacement of the carbonate. The result is a one-step synthesis of indolines which may be oxidized to indoles. The utility of the procedure is illustrated by the two- or three-step syntheses of anhydrolycorinone, hippadine, oxoassoanine, and pratosine.

2-Acylpyridazin-3-ones: Novel mild and chemoselective acylating agents for amines

2-Acyl-4,5-dichloropyridazin-3-ones served as excellent novel N-acylating reagents for amines under neutral conditions in organic solvent. They are convenient, chemoselective and easy to handle stable N-acylating reagents of amines.