36684-47-6

Upstream product

• 88-67-5 2-Iodobenzoic acid 
• 90-04-0 2-methoxy-phenylamine 
• 609-67-6 2-Iodobenzoyl chloride 

Downstream Products

• 106664-01-1 2-(2-methoxyphenyl)benzo[d][1,2]selenazol-3(2H)-one 
• 1628347-80-7 8-chloro-10-(2-methoxyphenyl)-5H-dibenzo[b,e][1,4]diazepin-11(10H)-one 
• 2314-77-4 N-(2-methoxyphenyl)phthalimide 
• 4299-25-6 2-(2-methoxyphenyl)benzo[d]isothiazol-3(2H)-one 
• 1402034-89-2 2,2'-selenobis(N-(2-methoxyphenyl)benzamide) 
• 3977-52-4 3-(2-methoxyphenyl)-4(3H)-quinazolinone 
• 934670-77-6 2-((4-aminophenyl)thio)-N-(2-methoxyphenyl)benzamide 
• 348132-55-8 N-(2-methoxyphenyl)-2-(phenylthio)benzamide 
• 431980-38-0 N-(2-methoxyphenyl)-2-((4-nitrophenyl)thio)benzamide 

Relevant academic research and scientific papers

PPh3/I2/HCOOH: An efficient CO source for the synthesis of phthalimides

A straightforward and general method has been developed for the synthesis of phthalimide derivatives from 2-iodobenzamides and PPh3/I2/HCOOH in the presence of a catalytic amount of Pd(OAc)2. The reaction results demonstrate that PPh3/I2/HCOOH is a facile, efficient and safe CO source. The whole process is carried out in toluene at 80 °C and furnishes the desired products in good to excellent yields.

Stable and Reusable Binaphthyl-Supported Palladium Catalyst for Aminocarbonylation of Aryl Iodides

A binaphthyl-supported Pd nanoparticles (Pd-BNP)-catalyzed aminocarbonylation of aryl iodides in the presence of carbon monoxide and amines for the synthesis of amides has been developed. This methodology provides an efficient route for the synthesis of a COX-2 enzyme inhibitor having anti-inflammatory activity.

Synthesis of dibenzodiazepinones via tandem copper(I)-catalyzed C-N bond formation

An efficient, one-pot method for the synthesis of dibenzodiazepinone derivatives involving copper-catalyzed tandem C-N bond formation is reported. The use of various halo amide and 2-iodoaniline derivatives permitted the synthesis of an array of dibenzodiazepinone derivatives in moderate to good yields. Moreover, a dibenzodiazepinone derivative {2-(11-oxo-5H-dibenzo[b,e][1, 4]diazepin-10(11H)-yl)benzonitrile} was utilized to synthesize the triazapentacyclic ring derivative {12-chloro- 8,15,22-triazapentacyclo[13.7.0. 02,7.09,14.016,21]docosa-1(22),2,4,6,9(14),10, 12,16(21),17,19-decaene}.

Composition and synthesis of new reagents for inhibition of HIV replication

The present invention provides compounds and compositions for inhibiting Vif and methods for treating viral infection, e.g., HIV infection.