367255-33-2Relevant academic research and scientific papers
Substituted indole-5-carboxamides and -acetamides as potent nonpeptide GnRH receptor antagonists
Ashton, Wallace T.,Sisco, Rosemary M.,Yang, Yi Tien,Lo, Jane-Ling,Yudkovitz, Joel B.,Cheng, Kang,Goulet, Mark T.
, p. 1723 - 1726 (2007/10/03)
The 2-aryltryptamine class of GnRH receptor antagonists has been modified to incorporate carboxamide and acetamide substituents at the indole 5-position. With either a phenol or methanesulfonamide terminus on the N-aralkyl side chain, potent binding affin
