402927-97-3

Basic information

• Product Name: 1-(METHYLSULFONYL)PIPERIDIN-4-AMINE
• Synonyms: ART-CHEM-BB B025717;1-(METHYLSULFONYL)PIPERIDIN-4-AMINE;AKOS B025717;4-Amino-N-1-(methylsulfonyl)piperidine;4-AMINO-1-METHANESULFONYLPIPERIDINE ;1-Methanesulfonyl-piperidin-4-ylamine;1-(methylsulfonyl)-4-piperidinamine(SALTDATA: HCl);1-(methylsulfonyl)-4-piperidinamine 1HCl
• CAS NO: 402927-97-3
• Molecular Formula: C₆H₁₄N₂O₂S
• Molecular Weight: 178.25
• Mol File: 402927-97-3.mol
• Article Data: 8

Chemical Properties

• Boiling Point: 296 °C at 760 mmHg
• Flash Point: 132.8 °C
• Appearance: /
• Density: 1.27 g/cm³
• Vapor Pressure: 0.00147mmHg at 25°C
• Refractive Index: 1.54
• Storage Temp.: Keep in dark place,Inert atmosphere,Room temperature
• PKA: 9.45±0.20(Predicted)
• CAS DataBase Reference: 1-(METHYLSULFONYL)PIPERIDIN-4-AMINE(CAS DataBase Reference)
• NIST Chemistry Reference: 1-(METHYLSULFONYL)PIPERIDIN-4-AMINE(402927-97-3)
• EPA Substance Registry System: 1-(METHYLSULFONYL)PIPERIDIN-4-AMINE(402927-97-3)

Safety Data

• Hazard Codes: Xi
• HazardClass: IRRITANT
• Hazardous Substances Data: 402927-97-3(Hazardous Substances Data)

Usage

General Description

1-(Methylsulfonyl)piperidin-4-amine is a chemical compound consisting of a piperidine ring with a sulfone group attached to the nitrogen atom. It is a stable, crystalline solid with a molecular formula of C9H19N3O2S. 1-(METHYLSULFONYL)PIPERIDIN-4-AMINE is commonly used in organic synthesis as a building block for the preparation of various pharmaceuticals and agrochemicals. It has shown potential as a starting material for the synthesis of antiviral and antitumor agents. Additionally, it has been studied for its potential use in the treatment of neurological disorders and as a precursor for the preparation of various biologically active compounds.

InChI:InChI=1/C6H14N2O2S/c1-11(9,10)8-4-2-6(7)3-5-8/h6H,2-5,7H2,1H3

Upstream product

• 402927-96-2 C₁₄H₂₀N₂O₄S 
• 73874-95-0 (piperidin-4-yl)carbamic acid tert-butyl ester 
• 287953-38-2 (1-methanesulfonyl-piperidin-4-yl)carbamic acid tert-butyl ester 

Downstream Products

• 1208147-14-1 C₂₄H₂₃Cl₂N₅O₃S 
• 741713-40-6 Ro 4584820 

Relevant articles and documents

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