40503-13-7Relevant academic research and scientific papers
Novel 4-(4-aryl)cyclohexyl-1-(2-pyridyl)piperazines as Δ8- Δ7 sterol isomerase (emopamil binding protein) selective ligands with antiproliferative activity
Berardi, Francesco,Abate, Carmen,Ferorelli, Savina,De Robertis, Anna F.,Leopoldo, Marcello,Colabufo, Nicola A.,Niso, Mauro,Perrone, Roberto
supporting information; experimental part, p. 7523 - 7531 (2009/12/07)
To find Δ8-Δ7 sterol isomerase (EBP) selective ligands, various arylpiperazines previously studied and structurally related to some σ receptors ligands were preliminarily screened. Consequently, a novel series of 2- or 2,6-disubstitu
