429669-07-8

Basic information

• Product Name: 1-BOC-3-(METHOXY)AZETIDINE
• Synonyms: 1-BOC-3-(METHOXY)AZETIDINE;1-Azetidinecarboxylicacid,3-methoxy-,1,1-dimethylethylester(9CI);3-Methoxy-azetidine-1-carboxylic acid tert-butyl ester;3-Methoxyazetidine, N-BOC protected;tert-Butyl 3-methoxyazetidine-1-carboxylate, 1-(tert-Butoxycarbonyl)-3-methoxyazetidine;tert-butyl 3-Methoxyazetidine-1-carboxylate;N-Boc-3-Methoxyazetidine;1-Azetidinecarboxylicacid, 3-Methoxy-, 1,1-diMethylethyl ester
• CAS NO: 429669-07-8
• Molecular Formula: C9H17NO3
• Molecular Weight: 187.23618
• Product Categories: METHOXY
• Mol File: 429669-07-8.mol
• Article Data: 10

Chemical Properties

• Boiling Point: 232.8±33.0 °C(Predicted)
• Appearance: /
• Density: 1.06±0.1 g/cm3(Predicted)
• Storage Temp.: Sealed in dry,Room Temperature
• PKA: -2.86±0.40(Predicted)
• CAS DataBase Reference: 1-BOC-3-(METHOXY)AZETIDINE(CAS DataBase Reference)
• NIST Chemistry Reference: 1-BOC-3-(METHOXY)AZETIDINE(429669-07-8)
• EPA Substance Registry System: 1-BOC-3-(METHOXY)AZETIDINE(429669-07-8)

Safety Data

• HazardClass: IRRITANT
• Hazardous Substances Data: 429669-07-8(Hazardous Substances Data)

Usage

General Description

1-BOC-3-(METHOXY)AZETIDINE is a specialized chemical compound that has a range of uses primarily in the field of chemistry and pharmaceuticals. Its molecular formula is C8H15NO3 and the molecular weight is 173.21 g/mol. This organic compound is a type of azetidine, a class of organic compounds featuring a four-membered ring structure containing three carbon atoms and one nitrogen atom. Specific information about its properties such as boiling point, melting point, density, or appearance may vary depending on the specific conditions under which the compound is handled or manipulated. Further details, including hazard identification and recommended safety measures, would be available on the chemical's Safety Data Sheet prepared by the manufacturer.

Upstream product

• 398489-26-4 tert-butyl 3-oxoazetidine-1-carboxylate 
• 74-88-4 methyl iodide 
• 24424-99-5 di-tert-butyl dicarbonate 
• 141699-55-0 tert-butyl 3-hydroxyazetidine-1-carboxylate 

Relevant articles and documents

Generation and electrophile trapping of N -Boc-2-lithio-2-azetine: Synthesis of 2-substituted 2-azetines

s-BuLi-induced α-lithiation-elimination of LiOMe from N-Boc-3-methoxyazetidine and further in situ α-lithiation generates N-Boc-2-lithio-2-azetine which can be trapped with electrophiles, either directly (carbonyl or heteroatom electrophiles) or after transmetalation to copper (allowing allylations and propargylations), providing a concise access to 2-substituted 2-azetines.

PDE9I WITH IMIDAZO PYRAZINONE BACKBONE

This invention is directed to compounds, which are PDE9 enzyme inhibitors. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of a compound of the invention and a pharmaceutically acceptable carrier. The pres

NEW BRADYKININ B1 ANTAGONISTS

The invention relates to compounds of formula (I) where in R1, R1a, R1b, R2, R3 and X, X1, X2, X3 have the meaning as cited in the description and the claims. Said compounds are useful as Bradykinin B1 antagonists. The invention also relates to pharmaceutical compositions, the preparation of such compounds as well as the production and use as medicament.