433953-62-9Relevant academic research and scientific papers
Synthesis of fluorescent biochemical tools related to the 2-azetidinone class of cholesterol absorption inhibitors
Burnett, Duane A.,Caplen, Mary Ann,Browne, Margaret E.,Zhau, Hongrong,Altmann, Scott W.,Davis Jr., Harry R.,Clader, John W.
, p. 315 - 318 (2002)
Fluorescent analogues of the cholesterol absorption inhibitor (CAI), Sch 58235, have been designed and synthesized as single enantiomers. Biological testing reveals that they are potent CAIs and are suitable tools for the investigation of the azetidinone CAI mechanism of action (MOA).
