446853-10-7Relevant academic research and scientific papers
Evaluation of diarylureas for activity against plasmodium falciparum
Zhang, Yiqun,Anderson, Marc,Weisman, Jennifer L.,Lu, Min,Choy, Cindy J.,Boyd, Vincent A.,Price, Jeanine,Sigal, Martina,Clark, Julie,Connelly, Michele,Zhu, Fangyi,Guiguemde, W. Armand,Jeffries, Cynthia,Yang, Lei,Lemoff, Andrew,Liou, Ally P.,Webb, Thomas R.,Derisi, Joseph L.,Guy, R. Kiplin
, p. 460 - 465 (2010)
A library of diarylurea insulin-like growth factor 1 receptor inhibitors was screened for activity against chloroquine-sensitive (3D7) and chloroquine-resistant (K1) strains of Plasmodium falciparum. The 4-aminoquinaldine-derived diarylureas displayed pro
