Evaluation of diarylureas for activity against plasmodium falciparum

DOI: 10.1021/ml100083c

Source and publish data:

ACS Medicinal Chemistry Letters p. 460 - 465 (2010)

Update date:2022-08-05

Topics:

Authors:

Zhang, Yiqun

Anderson, Marc

Weisman, Jennifer L.

Lu, Min Lu, Min

Choy, Cindy J.

Boyd, Vincent A.

Price, Jeanine

Sigal, Martina

Clark, Julie

Connelly, Michele

Zhu, Fangyi

Guiguemde, W. Armand

Jeffries, Cynthia

Yang, Lei

Lemoff, Andrew

Liou, Ally P.

Webb, Thomas R.

Derisi, Joseph L.

Guy, R. Kiplin

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Article abstract of DOI:10.1021/ml100083c

A library of diarylurea insulin-like growth factor 1 receptor inhibitors was screened for activity against chloroquine-sensitive (3D7) and chloroquine-resistant (K1) strains of Plasmodium falciparum. The 4-aminoquinaldine-derived diarylureas displayed pro

Full text of DOI:10.1021/ml100083c

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