4783-59-9Relevant academic research and scientific papers
HETEROARYL ARYL ETHERS
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Page/Page column 4, (2010/07/10)
The present invention relates to a process for the preparation of optionally substituted heteroaryl aryl ethers, in particular of phenoxypyridines.
Effect of microwave heating on Ullmann-type heterocycle-aryl ether synthesis using chloro-heterocycles
D'Angelo, Noel D.,Peterson, Joseph J.,Booker, Shon K.,Fellows, Ingrid,Dominguez, Celia,Hungate, Randall,Reider, Paul J.,Kim, Tae-Seong
, p. 5045 - 5048 (2007/10/03)
Ullmann ether synthesis was conducted on a variety of chloro-heterocycles with different phenols using optimized conditions involving copper powder and cesium carbonate. On many substrates, microwave heating afforded higher yields in significantly shorter reaction times compared to conventional heating conditions. These findings provide a facile method for aryl ether synthesis from chloropyridines, chloroquinolines, and chlorobenzothiazoles.
Oxamides as novel NR2B selective NMDA receptor antagonists
Barta-Szalai, Gizella,Borza, Istvan,Bozo, Eva,Kiss, Csilla,Agai, Bela,Proszenyak, Agnes,Keseru, Gyoergy M.,Gere, Aniko,Kolok, Sandor,Galgoczy, Kornel,Horvath, Csilla,Farkas, Sandor,Domany, Gyoergy
, p. 3953 - 3956 (2007/10/03)
A novel series of oxamides derived from indole-2-carboxamides was identified as potent NR2B selective NMDA receptor antagonists. Several members of this group showed good analgesic activity in the mouse formalin test.
