481630-71-1Relevant articles and documents
Advancing Base-Metal Catalysis: Development of a Screening Method for Nickel-Catalyzed Suzuki-Miyaura Reactions of Pharmaceutically Relevant Heterocycles
Goldfogel, Matthew J.,Guo, Xuelei,Gurak, John A.,Joannou, Matthew V.,Meléndez Matos, Jeishla L.,Moffat, William B.,Simmons, Eric M.,Wisniewski, Steven R.
supporting information, (2021/08/18)
Interest in replacing palladium catalysts with base metals resulted in the development of a 24-reaction screening platform for identifying nickel-catalyzed Suzuki-Miyaura reaction conditions. This method was designed to be directly applicable to process s
Structure-activity evaluation of n-benzyl-5-substituted indole-3-imine derivatives and their amine congeners as bovine testicular hyaluronidase (BTH) inhibitor
Oelgen,Kaessler,Kilic Kurt,Jose
experimental part, p. 685 - 690 (2012/04/05)
With the aim to overcome the lack of potent and selective Hyaluronidases (Hyals) inhibitors, we have tested new 1, 3 and 5 substituted indole derivatives for the inhibition of bovine testicular hyaluronidases (BTH) in a stains-all assay at pH 7 and in a M
Synthesis and pp60c-Src tyrosine kinase inhibitory activities of novel indole-3-imine and amine derivatives substituted at N1 and C5
Kilic, Zuhal,Isgoer, Yasemin G.,Oelgen, Suereyya
experimental part, p. 333 - 343 (2009/10/24)
A series of novel 1,3,5-trisubstituted indole derivatives, namely, N-benzyl 5-phenyl indole-3-imine, N-benzyl-5-(p-fluorophenyl)indole-3-imine and their corresponding amine congeners, were designed and synthesized as pp60 c-Src tyrosine kinase
