502545-86-0Relevant articles and documents
Structure-activity relationship study and drug profile of N-(4-fluorophenylsulfonyl)-L-valyl-L-leucinal (SJA6017) as a potent calpain inhibitor
Inoue, Jun,Nakamura, Masayuki,Cui, Ying-She,Sakai, Yusuke,Sakai, Osamu,Hill, Jeanette R.,Wang, Kevin K. W.,Yuen, Po-Wai
, p. 868 - 871 (2007/10/03)
Novel N-arylsulfonyldipeptidyl aldehyde derivatives were prepared by DMSO oxidation from the corresponding dipeptide alcohol, and their potencies as calpain inhibitors were evaluated in vitro. Among them, N-(4-fluorophenylsulfonyl)-L-valyl-L-leucinal (8,