50487-74-6Relevant articles and documents
Regio- and stereocontrolled synthesis of novel 3-sulfonamido-2,3,4,5- tetrahydro-1,5-benzothiazepines from 2-(bromomethyl)- or 2-(sulfonyloxymethyl) aziridines
Karikomi, Michinori,D'Hooghe, Matthias,Verniest, Guido,De Kimpe, Norbert
scheme or table, p. 1902 - 1904 (2009/01/31)
2-(Bromomethyl)-1-sulfonylaziridines were converted into novel 3-sulfonamido-2,3,4,5-tetrahydro-1,5-benzothiazepines upon treatment with 2-aminothiophenol in THF in the presence of K2CO3. Starting from 3-substituted 2-(sulfonyloxymet