509152-22-1Relevant academic research and scientific papers
Microwave promoted amination of 3-bromoisoxazoles
Moore, Jane E.,Spinks, Daniel,Harrity, Joseph P. A.
, p. 3189 - 3191 (2004)
This Letter describes the amination of 3-bromoisoxazoles by a nucleophilic aromatic substitution reaction. We have found 3-bromoisoxazoles to be inert to substitution under thermal conditions, however, the employment of phosphazene bases under microwave i
Synthesis of 3-haloisoxazole boronic esters: Novel heterocyclic synthetic intermediates containing independently variable functionality
Moore, Jane E.,Goodenough, Katharine M.,Spinks, Daniel,Harrity, Joseph P.A.
, p. 2071 - 2073 (2007/10/03)
The regioselective cycloaddition reaction of nitrile oxides with alkynylboronates has been exploited in the preparation of 3-bromo- and 3-chloroisoxazolyl-4-boronates. The synthetic potential of these intermediates has been explored through a number of cr
