5215-30-5Relevant academic research and scientific papers
Direct amide synthesis: via Ni-mediated aminocarbonylation of arylboronic acids with CO and nitroarenes
Shen, Ni,Cheung, Chi Wai,Ma, Jun-An
supporting information, p. 13709 - 13712 (2019/11/19)
Herein we describe an alternative and unconventional approach of an aminocarbonylation reaction to access aryl amides from readily available and low-cost arylboronic acids and nitroarenes. Nickel metal can serve as both reductant and catalyst in this direct aminocarbonylation. This protocol exhibits a good functional group compatibility and allows a variety of aryl amides to be synthesized, including several drug-like molecules.
Antimycobacterial activity of 3'- and 4'-fluorothiobenzanilides
Waisser,Kunes,Odlerova,Roman,Kubicova,Horak
, p. 193 - 195 (2007/10/03)
On the basis of a preliminary study of the antimycobacterial activity of thiobenzanilides, a group of 3/-fluoro- and 4/fluorothiobenzanilides has been synthesized and tested against Mycobacterium tuberculosis, M. kansasii, M. avium and M. fortuitum. The r
