53316-52-2Relevant academic research and scientific papers
2,4(5)-Diarylimidazoles as inhibitors of hNaV1.2 sodium channels: Pharmacological evaluation and structure-property relationships
Fantini, Marco,Rivara, Mirko,Zuliani, Valentina,Kalmar, Christopher L.,Vacondio, Federica,Silva, Claudia,Baheti, Aparna R.,Singh, Natasha,Merrick, Ellen C.,Katari, Ravi S.,Cocconcelli, Giuseppe,Ghiron, Chiara,Patel, Manoj K.
, p. 3642 - 3648 (2009)
Sodium (Na) channels continue to represent an important target for the development of novel anticonvulsants. We have synthesized and evaluated a series of 2,4(5)-diarylimidazoles for inhibition of the human neuronal NaV1.2 Na channel isoform. S
