58582-72-2Relevant academic research and scientific papers
2-Benzazepines. 5. Synthesis of pyrimido[5,4-d][2]benzazepines and their evaluation as anxiolytic agents
Trybulski, Eugene J.,Benjamin, Louis E.,Earley, James V.,Fryer, R. Ian,Gilman, Norman W.,et al.
, p. 1589 - 1596 (2007/10/02)
A series of 5H-pyrimido[5,4-d][2]benzazepines has been synthesized, starting from the corresponding 2-benzazepine-5-ones, and evaluated as potential anxiolytic agents. Selected compounds from this series show a pharmacological profile of action different
Pyrazolobenzazepines
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, (2008/06/13)
6-Aryl-1- or 2H,4H-pyrazolo[4,3-d](2)-benzazepines, e.g. those of the formula STR1 R = H or alkyl R° = H, alkyl, (HO, alkoxy, amino)-alkyl, aralkyl, aryl or acyl, R' = h, oh or alkyl R" = h, alkyl, alkoxy, halo or CF3 N-oxides thereof or therapeutically useful acid addition salts of such compounds exhibit antianxiety and antidepressant effects.
Pyrazolobenzazepines
-
, (2008/06/13)
6-Aryl-1- or 2H,4H-pyrazolo[4,3-d](2) -benzazepines, e.g. those of the formula STR1 N-oxides thereof or therapeutically useful acid addition salts of such compounds exhibit antianxiety and antidepressant effects.
