586412-27-3Relevant articles and documents
Discovery of potent, orally bioavailable, selective 5-HT1A/B/D receptor antagonists
Ward, Simon E.,Eddershaw, Peter J.,Scott, Claire M.,Gordon, Laurie J.,Lovell, Peter J.,Moore, Susan H.,Smith, Paul W.,Starr, Kathryn R.,Thewlis, Kevin M.,Watson, Jeannette M.
supporting information; experimental part, p. 2887 - 2890 (2009/04/11)
5-HT1 receptor antagonists have been discovered with good selectivity over the 5-HT transporter. This is the first report of highly potent, selective ligands for the 5-HT1A/B/D receptors with low intrinsic activity, which represent a
