634923-08-3Relevant academic research and scientific papers
Solution-phase synthesis of linear and cyclic peptidomimetics based on 2-aminoalkyloxazole-4- Or -5-carboxylates
Cox, Matthew O.,Prager, Rolf H.,Svensson, Carina E.
, p. 747 - 758 (2004)
The solution-phase synthesis of several small linear and cyclic peptidomimetics based on the coupling of BOC-protected 2-aminoalkyloxazole-4- or -5-carboxylic acids is reported. Cyclic amides have been formed both by sequential coupling and cyclization, o
The synthesis of some chiral 2-aminoalkyloxazole-5-carboxylates from isoxazol-5(2H)-ones
Cox, Matthew,Prager, Rolf H.,Svensson, Carina E.,Taylor, Max R.
, p. 897 - 901 (2007/10/03)
Ethyl 5-oxo-2,5-dihydroisoxazole-4-carboxylates have been N-acylated by a number of natural and synthetic phthalimidylamino acids in the presence of carbodiimides. The N-acylated products form the corresponding 2-aminoalkyloxazole-5-carboxylates smoothly when irradiated at 300 nm in acetone.
