6380-12-7Relevant academic research and scientific papers
Copper-catalyzed intermolecular C-H amination of (Hetero)arenes via transient unsymmetrical λ3-iodanes
Sokolovs, Igors,Lubriks, Dmitrijs,Suna, Edgars
supporting information, p. 6920 - 6928 (2014/06/09)
A one-pot two-step method for intermolecular C-H amination of electron-rich heteroarenes and arenes has been developed. The approach is based on a room-temperature copper-catalyzed regioselective reaction of the in situ formed unsymmetrical (hetero)aryl-λ3-iodanes with a wide range of primary and secondary aliphatic amines and anilines.
Synthesis, structural characterization and biological screening of various sulfa drugs derived from 2-anisidine
Abbasi, Muhammad Athar,Aziz-Ur-Rehman,Muhmood, Tahir,Khan, Khalid Mohammed,Ashraf, Muhammad,Ejaz, Syeda Abida,Arshad, Samreen
, p. 404 - 410 (2013/07/27)
In the present study, a series of N-alkyl substituted sulfa drugs (sulfonamides) has been synthesized. The reaction of 2-anisidine (1) with 4-methylbenzenesulfonyl chloride (2) yielded N- (2-methoxyphenyl)-4- methylbenzenesulfonamide (3), which on bromina
