639852-53-2Relevant academic research and scientific papers
Synthesis and evaluation as glycosidase inhibitors of carbasugar-derived spirodiaziridines, spirodiazirines, and spiroaziridines
Kapferer, Peter,Birault, Veronique,Poisson, Jean-Francois,Vasella, Andrea
, p. 2210 - 2227 (2007/10/03)
The spirodiaziridines 6 and 9, potential inhibitors of α- and β-glucosidases, were prepared from the validoxylamine A-derived cyclohexanone 5. The trimethylsilyl protecting groups of 5 are crucial for the formation of 6 in good yields. Oxidation of 6 gave
