683276-76-8Relevant academic research and scientific papers
Hydrophobic substituents on isatin derivatives enhance their inhibition against bacterial peptidoglycan glycosyltransferase activity
Chan, Kin-Fai,Chen, Yu Wai,Cheong, Wing-Lam,Liang, Zhiguang,So, Lok-Yan,So, Pui-Kin,Wang, Yong,Wong, Kwok-Yin,Wong, Wing-Leung
, (2020)
Moenomycin A, the well-known natural product inhibitor of peptidoglycan glycosyltransferase (PGT), is a large amphiphilic molecule of molecular mass of 1583 g/mol and its bioavailablity as a drug is relatively poor. In searching for small-molecule ligands
SSAO INHIBITOR
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Paragraph 0154; 0155; 0158; 0300; 0301; 0303, (2020/04/02)
The present invention provides an SSAO inhibitor and an application thereof in preparing a drug for treating a disease related to SSAO. In particular, the present invention provides a compound shown in formula (IV) and a pharmaceutically acceptable salt thereof.
3-IMINO-2-INDOLONES FOR THE TREATMENT OF DEPRESSION AND/OR ANXIETY
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, (2008/06/13)
This invention is directed to indolone derivatives which are selective antagonists for the GalR3 receptor. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of a compound of the invention and a pharmaceutica
3-Imino-2-indolones for the treatement of depression and/or anxiety
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, (2010/02/06)
This invention is directed to indolone derivatives which are selective antagonists for the GalR3 receptor. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of a compound of the invention and a pharmaceutica
