Bioorganic Chemistry (2020)
Update date:2022-08-04
Topics:
Chan, Kin-Fai
Chen, Yu Wai
Cheong, Wing-Lam
Liang, Zhiguang
So, Lok-Yan
So, Pui-Kin
Wang, Yong
Wong, Kwok-Yin
Wong, Wing-Leung
Moenomycin A, the well-known natural product inhibitor of peptidoglycan glycosyltransferase (PGT), is a large amphiphilic molecule of molecular mass of 1583 g/mol and its bioavailablity as a drug is relatively poor. In searching for small-molecule ligands
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