685134-51-4Relevant academic research and scientific papers
A solution-phase procedure for the preparation of 4-azasteroid mimetics
Ruda, Marcus C.,Bergman, Jan,Koehler, Konrad,Liu, Ye
, p. 571 - 574 (2003)
A Diels-Alder approach has been employed to make 3-oxo-octahydro-benzo[f] quinoline derivatives as ligands for nuclear hormone receptors and steroid biosynthetic enzymes. The five-step synthesis is a model for the synthesis of libraries on solid-phase.
NOVEL NUCLEAR HORMONE RECEPTOR LIGANDS AND METHODS
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Page 22-23, (2008/06/13)
The present invention relates to compounds and derivatives thereof, their synthesis, and their use as nuclear hormone receptor modulators. The compounds of the instant invention are ligands for nuclear hormone receptors and as such may be useful for treat
