72360-04-4Relevant academic research and scientific papers
Discovery of orally available 8-aza-5-thiaProstaglandin E1 analogs as highly selective EP4 agonists
Kambe, Tohru,Maruyama, Toru,Nakano, Masayuki,Yamaura, Yoshiyuki,Shono, Tomoyuki,Seki, Akiteru,Sakata, Kiyoto,Maruyama, Takayuki,Nakai, Hisao,Toda, Masaaki
, p. 1523 - 1534 (2012/01/13)
Analogs 8-aza-16-aryl prostaglandin E1 (PGE1) and 8-aza-5-thia-16-arylPGE1 were synthesized and evaluated with respect to their subtype receptor affinity and EP4 agonist activity for the purposes of identifying sub-type- selective EP
Cyclic ketone derivatives and their medical applications
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, (2008/06/13)
The present invention relates to cyclic ketones represented by the following formula and to drugs in which an effective component is such a cyclic ketone or a pharmacologically acceptable salt thereof.The cyclic ketones of the present invention encourage the production of blood platelets, leukocytes and erythrocytes, and can be employed in the prevention or treatment of cytopaenia brought about by cancer chemotherapy, radiotherapy or drug therapy, or by immunological abnormality, anaemia and the like.
Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands
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, (2008/06/13)
PCT No. PCT/GB94/01936 Sec. 371 Date Mar. 12, 1996 Sec. 102(e) Date Mar. 12, 1996 PCT Filed Sep. 6, 1994 PCT Pub. No. WO95/07893 PCT Pub. Date Mar. 23, 1995A class of fused tricyclic heteroaromatic compounds of formula (I) as defined in claim 1 or a salt
LONG-ACTING CONTRACEPTIVE AGENTS: LEVONORGESTREL ESTERS OF UNSATURATED ACIDS
Wan, A. S. C.,Ngiam, T. L.,Leung, S. L.,Go, M. L.,Francisco, C. G.,et al.
, p. 339 - 348 (2007/10/02)
Esters of levonorgestrel (13β-ethyl-17α-ethynyl-17β-hydroxygon-4-en-3-one) with a variety of unsaturated carboxylic acids have been synthesized for evaluation as potential long-acting, injectable contraceptive agents.
