752986-14-4Relevant academic research and scientific papers
2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists
Scheiff, Anja B.,Yerande, Swapnil G.,El-Tayeb, Ali,Li, Wenjin,Inamdar, Gajanan S.,Vasu, Kamala K.,Sudarsanam, Vasudevan,Müller, Christa E.
experimental part, p. 2195 - 2203 (2010/06/12)
A series of 2-amino-5-benzoyl-4-phenylthiazole derivatives was investigated in radioligand binding studies at adenosine receptor (AdoR) subtypes with the goal to obtain potent and A1-selective antagonists. Acylation of the 2-amino group was fou
