761374-82-7Relevant articles and documents
Synthesis of 4-Substituted 11-Phenyl-1,2,3,4-tetrahydro-5H-azepinoquinolin-5-one Derivatives as Potential Peripheral Benzodiazepine-Receptor Ligands
Cappelli, Andrea,Anzini, Maurizio,Vomero, Salvatore
, p. 1265 - 1272 (2007/10/02)
The synthesis of semirigid analogs of PK 11195, the highly specific peripheral benzodiazepine-receptor ligand, is reported.Compound (4) underwent the Wittig reaction with acetaldehyde to give olefin (7) which after allylic bromination was aminated to give