766547-97-1Relevant academic research and scientific papers
SAR and pharmacokinetic studies on phenethylamide inhibitors of the hepatitis C virus NS3/NS4A serine protease
Malancona, Savina,Colarusso, Stefania,Ontoria, Jesus M.,Marchetti, Antonella,Poma, Marco,Stansfield, Ian,Laufer, Ralph,Di Marco, Annalise,Taliani, Marina,Verdirame, Maria,Gonzalez-Paz, Odalys,Matassa, Victor G.,Narjes, Frank
, p. 4575 - 4579 (2007/10/03)
SAR on the phenethylamide 1 (Ki 1.2μM) in the P2- and the P′-position led to potent inhibitors, one of which showed good exposure and low clearance when administered intramuscularly to rat.
