77893-68-6Relevant articles and documents
2-AMINO-N-(AMINO-OXO-ARYL-LAMBDA6-SULFANYLIDENE)ACETAMIDE COMPOUNDS AND THEIR THERAPEUTIC USE
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Page/Page column 222, (2021/06/26)
The present invention pertains generally to the field of therapeutic compounds. More specifically the present invention pertains to certain 2-amino-N-(amino-oxo-aryl-λ6- sulfanylidene)acetamide compounds (referred to herein as ANASIA compounds) that, inter alia, inhibit (e.g., selectively inhibit) bacterial aminoacyl-tRNA synthetase (aaRS) (e.g., bacterial leucyl-tRNA synthetase, LeuRS). The present invention also pertains to pharmaceutical compositions comprising such compounds, and the use of such compounds and compositions, both in vitro and in vivo, to inhibit (e.g., selectively inhibit) bacterial aminoacyl-tRNA synthetase; to treat disorders that are ameliorated by the inhibition (e.g., selective inhibition) of bacterial aminoacyl-tRNA synthetase; to treat bacterial infections; etc.
CYCLIC SULFAMIDE COMPOUNDS AND METHODS OF USING SAME
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Page/Page column 309, (2018/09/21)
The present disclosure provides, in part, cyclic sulfamide compounds, and pharmaceutical compositions thereof, useful as modulators of Hepatitis B (HBV) core protein, and methods of treating Hepatitis B (HBV) infection.
PRODUCTION METHOD OF DITHIENOBENZODITHIOPHENE
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Paragraph 0047, (2016/12/01)
PROBLEM TO BE SOLVED: To provide an efficient production method of dithienobenzodithiophene and its derivatives which imparts high carrier mobility by application and enables easy and efficient film production of an organic semiconductor layer. SOLUTION: A production method of dithienobenzodithiophene is characterized by producing dithienobenzodithiophene by using 2,3-dihalothiophene whose halogen at 2-position is equal in atomic number to, or larger than, the halogen at 3-position. COPYRIGHT: (C)2016,JPOandINPIT