813447-29-9Relevant academic research and scientific papers
N-[(3S)-Pyrrolidin-3-yl]benzamides as novel dual serotonin and noradrenaline reuptake inhibitors: Impact of small structural modifications on P-gp recognition and CNS penetration
Wakenhut, Florian,Allan, Gill A.,Fish, Paul V.,Jonathan Fray,Harrison, Anthony C.,McCoy, Rachel,Phillips, Stephen C.,Stobie, Alan,Westbrook, Dominique,Westbrook, Simon L.,Whitlock, Gavin A.
scheme or table, p. 5078 - 5081 (2010/03/24)
The structure-activity relationship and the synthesis of novel N-[(3S)-pyrrolidin-3-yl]benzamides as dual serotonin and noradrenaline monoamine reuptake inhibitors (SNRI) is described. Preferred compound 9 aka PF-184,298 is a potent SNRI with good selecti
N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS SEROTONIN AND NORADRENALINE RE-UPTAKE INHIBITORS
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Page 44, (2008/06/13)
A compound of Formula (I) and pharmaceutically and/or veterinarily acceptable derivatives thereof, wherein R1 is H, C1_6alkyl, -C(X)Y, C3_8cycloalkyl, aryl, het, aryl-Cl_4alkyl o
