83160-06-9Relevant academic research and scientific papers
Synthesis and Pharmacological Characterization in Vitro of Cyclic Enkephalin Analogues: Effect of Conformational Constraints on Opiate Receptor Selectivity
DiMaio, John,Nguyen, Thi M.-D.,Lemieux, Carole,Schiller, Peter W.
, p. 1432 - 1438 (2007/10/02)
Using a combination of solid-phase and solution methods, we synthesized a series of cyclic 5> enkephalin analogues by substitution of D-α,ω-diamino acids in position 2 of the enkephalin sequence and cyclization of the ω-amino group to the C
