83283-25-4Relevant academic research and scientific papers
Thioamides: Synthesis, stability, and immunological activities of thioanalogues of imreg. Preparation of new thioacylating agents using fluorobenzimidazolone derivatives
Zacharie, Boulos,Lagraoui, Mouna,Dimarco, Marika,Penney, Christopher L.,Gagnon, Lyne
, p. 2046 - 2052 (2007/10/03)
Imreg (Tyr1-Gly2-Gly3) is a well-known immunostimulant. However, it possesses a short half-life. Stabilized analogues of Imreg were prepared by a regioselective insertion in which peptide bonds at position 1,2 or 2,3 were
ENDOTHIOPEPTIDES
Brown, D. W.,Campbell, M. M.,Walker, C. V.
, p. 1075 - 1083 (2007/10/02)
N-protected dipeptide esters have been converted into the corresponding protected endothiopeptides using Lawesson's reagent, 1.Methods of amino and carboxyl deprotection, and coupling of the thiopeptides with amino acids have been defined and used to prep
