836633-05-7Relevant academic research and scientific papers
Scaffold oriented synthesis. Part 1: Design, preparation, and biological evaluation of thienopyrazoles as kinase inhibitors
Akritopoulou-Zanze, Irini,Darczak, Daria,Sarris, Kathy,Phelan, Kathleen M.,Huth, Jeffrey R.,Song, Danying,Johnson, Eric F.,Jia, Yong,Djuric, Stevan W.
, p. 96 - 99 (2007/10/03)
We report the synthesis of kinase targeted libraries based on the thienopyrazole scaffold. Several thienopyrazole analogs have been identified as submicromolar inhibitors of KDR.
Substituted thieno [2,3-c] pyrazoles and their use as medicinal products
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Page 6, (2008/06/13)
The present invention relates in particular to novel chemical compounds, particularly novel substituted thieno[2,3-c]pyrazoles, to the compositions containing them and to their use as medicinal products for treating cancers and also neurodegenerative dise
