849935-46-2Relevant academic research and scientific papers
Novel acetylcholinesterase inhibitor as increasing agent on rhythmic bladder contractions: SAR of 8-{3-[1-(3-fluorobenzyl)piperidin-4-yl]propanoyl}- 1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one (TAK-802) and related compounds
Ishichi, Yuji,Sasaki, Mitsuru,Setoh, Masaki,Tsukamoto, Tetsuya,Miwatashi, Seiji,Nagabukuro, Hiroshi,Okanishi, Satoshi,Imai, Shigemitsu,Saikawa, Reiko,Doi, Takayuki,Ishihara, Yuji
, p. 1901 - 1911 (2007/10/03)
As part of an on-going investigation to develop an increasing agent on rhythmic bladder contractions, 1-aryl-3-(1-benzylpiperidin-4-yl)propanones were synthesized and examined as noncarbamate acetylcholinesterase (AChE) inhibitors. Among compounds with va
