85126-66-5Relevant academic research and scientific papers
Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin- 2-yl)-4-(quinolin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors
Jin, Cheng Hua,Krishnaiah, Maddeboina,Sreenu, Domalapally,Rao, Kota Sudhakar,Subrahmanyam, Vura Bala,Park, Chul-Yong,Son, Jee-Yeon,Sheen, Yhun Yhong,Kim, Dae-Kee
experimental part, p. 2633 - 2640 (2011/06/11)
A series of 1-substituted-3(5)-(6-methylpyridin-2-yl)-4-(quinolin-6-yl) pyrazoles 14a-e, 15a-e, 17a-c, and 18a-d have been synthesized and evaluated for their ALK5 inhibitory activity in an enzyme assay and in a cell-based luciferase reporter assay. The 6
Substituted benzamide radiosensitizers
-
, (2008/06/13)
A method for sensitizing hypoxic tumor cells to radiation using derivatives of benzamide are disclosed. Some of the compounds useful in the REFERENCE TO GOVERNMENT GRANT OR CONTRACT The invention described herein was made in the course of work under grant or contract from the National Institutes of Health.
