861306-84-5Relevant articles and documents
Antiprotozoal activity and DNA binding of dicationic acridones
Montalvo-Quirós, Sandra,Taladriz-Sender, Andrea,Kaiser, Marcel,Dardonville, Christophe
, p. 1940 - 1949 (2015/04/21)
Dicationic acridone derivatives were synthesized and their antiparasitic activity was evaluated. Acridones displayed in vitro nanomolar IC50 values against Trypanosoma brucei rhodesiense STIB900 with selectivity indices >1000. Compounds 1b, 3a,