864296-43-5Relevant academic research and scientific papers
3-AMINO-INDAZOLE OR 3-AMINO-4,5,6,7-TETRAHYDRO-INDAZOLE DERIVATIVES
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Page/Page column 19, (2010/04/23)
This invention relates to novel indazole derivatives of formula I: wherein R1 to R7 are as defined in the description and in the claims, as well as physiologically acceptable salts thereof. These compounds are FXR modulators and can
Benzoylurea oligomers: Synthetic foldamers that mimic extended α helices
Rodriguez, Johanna M.,Hamilton, Andrew D.
, p. 8614 - 8617 (2008/09/18)
Not-so-short and curlies: A new benzoylurea-based foldamer scaffold favors a linear conformation governed by intramolecular hydrogen bonding (see picture, left). The functional groups R are in a staggered arrangement analogous to an α helix. Iterative syn
New carboxylic acid amides, the preparation thereof and their use as medicaments
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Page/Page column 48, (2010/02/13)
The present invention relates to new substituted carboxylic acid amides of general formula wherein A, B and R1 to R5 are defined as in claim 1, the tautomers, the enantiomers, the diastereomers, the mixtures thereof and the salts thereof, particularly the physiologically acceptable salts thereof with inorganic or organic acids or bases, which have valuable properties.
NOVEL CARBOXAMIDES FOR USE AS XA INHIBITORS
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Page/Page column 124-125, (2010/02/13)
The invention relates to the novel substituted carboxamides of general formula (I), wherein A, B and R1 to R5 are defined as in claim 1, the tautomers, enantiomers, diastereomers, mixtures and salts thereof, especially the physiologically salts thereof with inorganic or organic acids or bases, which have valuable properties. The inventive compounds have an antithrombotic effect and are factor Xa inhibitors.
