865444-78-6Relevant articles and documents
Bromine structural domain inhibitor compound and application thereof
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Paragraph 0135-0136; 0139-0140, (2019/08/02)
The invention relates to a bromine structural domain inhibitor and provides a compound shown in a general formula I, pharmaceutical salt, an enantiomer, a diastereoisomer, an atropisomer, racemate, apolymorphic substance and solvate of the compound or an isotope labelled compound (including a deuterium substituted compound), a preparation method of the compound, pharmaceutical composition containing the compound and an application of the above components in pharmaceuticals.
NEW TRPA1 ANTAGONISTS
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Page/Page column 55, (2017/08/01)
The present invention relates to compounds of Formula (I), to the process for preparing such compounds and to their use in the treatment of a pathological condition or disease susceptible to amelioration by TRPA1 channel inhibition or antagonism.
Methods for synthesizing imidazotriazinones
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Page/Page column 8; 9, (2008/06/13)
Methods of synthesizing imidazotriazinones, such as vardenafil, and compositions useful for the same are disclosed.