869012-93-1Relevant academic research and scientific papers
Practical regioselective bromination of azaindoles and diazaindoles
Gallou, Fabrice,Reeves, Jonathan T.,Tan, Zhulin,Song, Jinhua J.,Yee, Nathan K.,Harcken, Christian,Liu, Pingrong,Thomson, David,Senanayake, Chris H.
, p. 211 - 214 (2007/10/03)
A mild and efficient synthesis of various 3-brominated azaindoles and diazaindoles was developed by regioselective halogenation of the parent systems. This practical and high-yielding transformation was achieved with copper(II) bromide in acetonitrile at
Regioselective halogenation of 6-azaindoles: Efficient synthesis of 3-halo-2,3-disubstituted-6-azaindole derivatives
Gallou, Fabrice,Reeves, Jonathan T.,Tan, Zhulin,Song, Jinhua J.,Yee, Nathan K.,Campbell, Scot,Jones, Paul-James,Senanayake, Chris H.
, p. 2400 - 2402 (2007/10/03)
A mild and efficient synthesis of 3-halo-2-substituted-6-azaindoles was developed by regioselective halogenation of 6-azaindole systems. The transformation was achieved with copper(II) bromide in acetonitrile at room temperature. Georg Thieme Verlag Stutt
