873211-41-7Relevant academic research and scientific papers
Magnesium dicarboxylates promote the prenylation of phenolics that is extended to the total synthesis of icaritin
Fu, Xuewen,Lu, Xiaoxia,Wang, Chun,Wen, Yongju,Xiong, Wei,Zhang, Guolin,Zhang, Jichao
, p. 1117 - 1124 (2022/02/16)
The prenylation of phenolic substrates promoted by magnesium dicarboxylates was developed. An investigation of the scope demonstrated that substrates with electron-donating group(s) gave better yields than those with electron-withdrawing group(s). Althoug
Design, Synthesis, and Structure–Activity Relationships of Bavachinin Analogues as Peroxisome Proliferator-Activated Receptor γ Agonists
Du, Guoxin,Zhao, Yuanyuan,Feng, Li,Yang, Zhuo,Shi, Jiye,Huang, Cheng,Li, Bo,Guo, Fujiang,Zhu, Weiliang,Li, Yiming
, p. 183 - 193 (2017/02/05)
Peroxisome proliferator-activated receptor γ (PPARγ) agonists have been used for the treatment of diabetes with the effect of lowering blood glucose levels and improving insulin sensitivity. Natural compounds such as flavones, flavanones, and isoflavones
Synthesis of?compounds with antiproliferative activity as?analogues of?prenylated natural products existing in?Brazilian propolis
Pisco, Laura,Kordian, Marcus,Peseke, Klaus,Feist, Holger,Michalik, Dirk,Estrada, Ernesto,Carvalho, Jo?o,Hamilton, Gerhard,Rando, Daniela,Quincoces, Jose
, p. 401 - 407 (2007/10/03)
This work describes the syntheses and antitumoral properties of five prenyl compounds from which antiproliferative activities were predicted by using the TOPS-MODE approach, a computational method for drug design. The syntheses of 2-(3-methylbut-2-enyloxy
SUBSTITUTED HYDROXYACETOPHENON DERIVATIVES
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Page/Page column 11; 12-13, (2008/06/13)
The invention relates to substituted hydroxyacetophenon derivatives having antiproliferative and antimicrobial properties, to medicaments containing said derivatives, and to a method for the production thereof. Furthermore, the inventive hydroxyacetopheno
Bismuth triflate catalyzed [1,3] rearrangement of aryl 3-methylbut-2-enyl ethers
Ollevier, Thierry,Mwene-Mbeja, Topwe M.
, p. 3963 - 3966 (2008/03/11)
An efficient bismuth triflate catalyzed [1,3] rearrangement of aryl 3-methylbut-2-enyl ethers has been developed. The reaction proceeds rapidly and affords the corresponding para- and ortho-prenylated phenols and naphthols in moderate to good yields (up t
