874278-18-9Relevant academic research and scientific papers
Small molecule antagonists of the gonadotropin-releasing hormone (GnRH) receptor: Structure-activity relationships of small heterocyclic groups appended to the 2-phenyl-4-piperazinyl-benzimidazole template
Hauze, Diane B.,Chengalvala, Murty V.,Cottom, Joshua E.,Feingold, Irene B.,Garrick, Lloyd,Green, Daniel M.,Huselton, Christine,Kao, Wenling,Kees, Kenneth,Lundquist IV, Joseph T.,Mann, Charles W.,Mehlmann, John F.,Rogers, John F.,Shanno, Linda,Wrobel, Jay,Pelletier, Jeffrey C.
scheme or table, p. 1986 - 1990 (2009/11/30)
A previous report described the serum LH suppression pharmacology of the 2-phenyl-4-piperazinyl-benzimidazole N-ethyluracil GnRH receptor antagonist 1 following oral administration in rats. A series of small heterocycles were appended to the 2-(4-tert-but
