879485-07-1Relevant academic research and scientific papers
3-(2-(AMINOETHYL)-INDOL-4-OL DERIVATIVES, METHODS OF PREPARATION THEREOF, AND THE USE AS 5-HT2 RECEPTOR MODULATORS
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, (2021/09/17)
A compound of Formula I, which possesses 5-HT2A and/or 5-HT2c selective receptor activity, but lacks at least some of the undesirable characteristics of 5-HT2B-agonist related activities, is disclosed. Methods of preparing said compo
SAR of psilocybin analogs: Discovery of a selective 5-HT2C agonist
Sard, Howard,Kumaran, Govindaraj,Morency, Cynthia,Roth, Bryan L.,Toth, Beth Ann,He, Ping,Shuster, Louis
, p. 4555 - 4559 (2007/10/03)
An SAR study of psilocybin and psilocin derivatives reveals that 1-methylpsilocin is a selective agonist at the h5-HT2C receptor. The corresponding phosphate derivative, 1-methylpsilocybin, shows efficacy in an animal model for obsessive-compul
